Name | CDK12-IN-4 | CAS# | 2651196-69-7 | |
---|---|---|---|---|
Price | ¥Inquiry/100mg ¥Inquiry/250mg ¥Inquiry/1g | Purity | 98.0% | |
Stocking Period |
1 Day | Stock | 3 | |
Product Webpage: | https://www.dcchemicals.com/product_show-cdk12-in-4.html |
Detail
Product Information
CDK12-IN-4, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC50 of 0.641 μM at high ATP (2 mM). CDK12-IN-4 has no effect on CDK2/Cyclin E (IC50>20 μM) and CDK9/Cyclin T1 (IC50>20 μM) at high ATP (2 mM) (WO2021116178A1). |