常用名 | CDK12-IN-4 | CAS号 | 2651196-69-7 |
---|---|---|---|
价格 | ¥需询单/100mg ¥需询单/250mg ¥需询单/1g | 纯度 | 98.0% |
备货期 | 1天 | 库存 | 3 |
产品网页 | https://www.dcchemicals.com/product_show-cdk12-in-4.html |
产品详情(用途,包装等)
CDK12-IN-4, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC50 of 0.641 μM at high ATP (2 mM). CDK12-IN-4 has no effect on CDK2/Cyclin E (IC50>20 μM) and CDK9/Cyclin T1 (IC50>20 μM) at high ATP (2 mM) (WO2021116178A1). |