Cobalt??Catalyzed Electrophilic Amination of Arylzincs with N??Chloroamines

…, Z Yu, A Auffrant, C Gosmini

Index: Qian, Xin; Yu, Zailu; Auffrant, Audrey; Gosmini, Corinne Chemistry - A European Journal, 2013 , vol. 19, # 20 p. 6225 - 6229

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Citation Number: 22

Abstract

Aromatic CÀN bond-forming reactions are important for the synthesis of biologically-active substructures and medicinal-chemistry targets.[1] Over the past decade, the Buchwald– Hartwig amination of electrophilic aromatics involving Pd,[2] Cu,[3] and Ni [4] centers has become a prominent and elegant method for creating CÀN bonds and forming functionalized arylamines. More recently, catalytic systems based on cobalt have also ...

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