Synthesis and biological activities of novel aryl indole-2-carboxylic acid analogs as PPARγ partial agonists

JF Dropinski, T Akiyama, M Einstein…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 15, # 22 p. 5035 - 5038

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Citation Number: 52

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... A medicinal chemistry effort was initiated based on the interesting biological profile of compound 1a ... The latter was converted to compounds 33–39 using either the previously discussed copper coupling or halide displacement chemistry. ...

Bausteine und Organisationsformen des Bindegewebes

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[Hickman; Sturino; Lachance Tetrahedron Letters, 2000 , vol. 41, # 43 p. 8217 - 8220]

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[Justus Liebigs Annalen der Chemie, , vol. 393, p. 358 Justus Liebigs Annalen der Chemie, , vol. 408, p. 280 DE105495 ; Fortschr. Teerfarbenfabr. Verw. Industriezweige, vol. 5, p. 400 Justus Liebigs Annalen der Chemie, , vol. 301, p. 350 Chem. Zentralbl., , vol. 71, # I p. 272 Chemische Berichte, , vol. 35, p. 1685]

Synthesis and biological activities of novel aryl indole-2-c...

[Dropinski, James F.; Akiyama, Taro; Einstein, Monica; Habulihaz, Bahanu; Doebber, Tom; Berger, Joel P.; Meinke, Peter T.; Shi, Guo Q. Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 22 p. 5035 - 5038]