2-Arylpropionic CXC chemokine receptor 1 (CXCR1) ligands as novel noncompetitive CXCL8 inhibitors

…, R Bertini, MC Cesta, C Bizzarri…

Index: Higgins, Stanley D.; Thomas, Barry C. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1982 , p. 235 - 242

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Citation Number: 92

Abstract

... Journal of Medicinal ... 2005, 48 (13), pp 4312–4331. DOI: 10.1021/jm049082i. Publication Date (Web): May 27, 2005. Copyright © 2005 American Chemical Society. ... wild-type CXCR1/L1.2 and mutated Lys99Ala CXCR1 cell membranes were incubated with [ 14 C]-1 and irradiated ...

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