Synthetic communications

Highly diastereoselective alkylation of the Dellaria oxazinone template with bifunctional electrophiles

GHP Roos, KA Dastlik

Index: Roos, Gregory H. P.; Dastlik, Kim A. Synthetic Communications, 2003 , vol. 33, # 13 p. 2197 - 2208

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Citation Number: 7

Abstract

Abstract This study investigates the efficiency of alkylation of the Dellaria oxazinone glycinate template with sensitive bifunctional electrophiles. In addition to improved access to the template, triflate/halide bifunctional combinations provided good yields (85–93%) of