Synthesis and quantitative structure–activity relationship (QSAR) study of novel N-arylsulfonyl-3-acylindole arylcarbonyl hydrazone derivatives as nematicidal agents

…, L Fan, H Xu, X Yu, X Zhi, X Yao, R Zhang

Index: Che, Zhiping; Zhang, Shaoyong; Shao, Yonghua; Fan, Lingling; Xu, Hui; Yu, Xiang; Zhi, Xiaoyan; Yao, Xiaojun; Zhang, Rui Journal of Agricultural and Food Chemistry, 2013 , vol. 61, # 24 p. 5696 - 5705

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Citation Number: 19

Abstract

In continuation of our program aimed at the discovery and development of natural-product- based pesticidal agents, 54 novel N-arylsulfonyl-3-acylindole arylcarbonyl hydrazone derivatives were prepared, and their structures were well characterized by 1H NMR, 13C NMR, HRMS, ESI-MS, and mp. Their nematicidal activity was evaluated against that of the pine wood nematode, Bursaphelenchus xylophilus in vivo. Among all of the derivatives, ...