Letters in Organic Chemistry

A Simple and Efficient Method for Trifluoroacetylation of Arylamines Using Trifluoroacetic Acid and Triphosgene

KJ Han, M Kim

Index: Han, Ki-Jong; Kim, Misoo Letters in Organic Chemistry, 2011 , vol. 8, # 8 p. 559 - 561

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Abstract

A simple and efficient one-pot procedure for trifluoroacetylation of arylamines using trifluoroacetic acid and triphosgene is reported. A mixed trifluoroacetic anhydride generated in situ reacts with a variety of arylamines to give the corresponding trifluroacetamides in high

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