Tetrahedron Letters

A versatile and efficient process to 3-substituted indoles from anilines

W Wierenga, J Griffin, MA Warpehoski

Index: Wierenga, Wendell; Griffin, John; Warpehoski, Martha A. Tetrahedron Letters, 1983 , vol. 24, # 24 p. 2437 - 2440

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Citation Number: 28

Abstract

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Borane-mediated reductive elimination of α-thiomethyl-, α-hydroxy, or α-alkoxy-, α′-substituted oxindoles affords 3-substituted indoles in high yield. Isatins, available several routes from oxindoles, also afford indoles. ... Gassman and van Bergen reported the reduction of 3- ...

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