Tetrahedron

(1-Bromovinyl)-MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis

EM Woerly, JE Miller, MD Burke

Index: Woerly, Eric M.; Miller, Jonathan E.; Burke, Martin D. Tetrahedron, 2013 , vol. 69, # 36 p. 7732 - 7740

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Citation Number: 11

Abstract

Abstract Iterative cross-coupling represents a potentially general approach for the simple, efficient, and flexible construction of a wide range of functional small molecules. In this context,(1-bromovinyl)-N-methyliminodiacetic acid (MIDA) boronate is a very useful building block for small molecule synthesis. This compound can serve as a starting material for the preparation of a wide range of 1, 1-disubstituted olefin-containing MIDA boronates. This ...