Facile and efficient carboalkoxylation and carboaryloxylation of amines

…, J Haruta, H Tagawa, Y Tamura

Index: Kita, Yasuyuki; Haruta, Jun-ichi; Tagawa, Hiroko; Tamura, Yasumitsu Journal of Organic Chemistry, 1980 , vol. 45, # 22 p. 4519 - 4522

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Citation Number: 25

Abstract

were done by the use of 3 equiv of 3a. Although we have not as yet investigated the limitations imposed on the reaction by the presence of other functional groups in detail, weakly basic groups such as the hydroxyl group, were found not to cause interference. Thus, an amino alcohol readily reacts with 3a to give the corresponding N-carboethoxylated compound as the sole product in a high yield. As indicated in Table I, the conditions were ...