Synthesis, biological testing, and stereochemical assignment of an end group modified retro-inverso bombesin C-terminal nonapeptide

M Cushman, J Jurayj, JD Moyer

Index: Cushman, Mark; Jurayj, Jurjus; Moyer, James D. Journal of Organic Chemistry, 1990 , vol. 55, # 10 p. 3186 - 3194

Full Text: HTML

Citation Number: 27

Abstract

The end group modified retro-inverso bombesin C-terminal nonapeptide 3 and its diastereomer 4 have been synthesized. The absolute configurations at the substituted malonamic acid residues in 3 and 4 were determined by chemical correlation with D-and L-2- aminobutyric acids of known absolute configuration. Thus, the absolute configurations at the substituted malonamic acid residues in each diastereomer of 25a were determined by ...

~99%

Total synthesis of the cyclic peptide argyrin B

[Ley, Steven V.; Priour, Alain European Journal of Organic Chemistry, 2002 , # 23 p. 3995 - 4004]

Highly practical methodology for the synthesis of d-and l-α-...

[Myers, Andrew G.; Gleason, James L.; Yoon, Taeyoung; Kung, Daniel W. Journal of the American Chemical Society, 1997 , vol. 119, # 4 p. 656 - 673]