HS024

• 常用名: HS024
• 英文名: Acetyl-(Cys3,Nle4,Arg5,D-2-Nal7,Cys11)-α-MSH (3-11) amide trifluoroacetate salt
• CAS号: 212370-59-7
• 分子量: 1266.499
• 密度: 1.5±0.1 g/cm3
• 沸点: N/A
• 分子式: C₅₈H₇₉N₁₉O₁₀S₂
• 熔点: N/A
• 闪点: N/A

HS024用途

HS024 is a selective MC4 receptor antagonist, with Kis of 0.29, 3.29, 5.45, and 18.6 nM for MC4, MC5, MC3, and MC1, respectively. HS024 increase food intake.

HS024名称

• 英文名: hs 024

HS024物理化学性质

• 密度: 1.5±0.1 g/cm3
• 分子式: C₅₈H₇₉N₁₉O₁₀S₂
• 分子量: 1266.499
• 精确质量: 1265.569824
• PSA: 550.86000
• LogP: -1.57
• 折射率: 1.717

HS024英文别名

• M.W. 1266.50 C58H79N19O10S2
• Neurodazine
• 1,2-Dithia-5,8,11,14,17,20,23,26-octaazacyclononacosane-4-carboxamide, 28-(acetylamino)-13,22-bis[3-[[(E)-aminoiminomethyl]amino]propyl]-25-butyl-19-(1H-imidazol-4-ylmethyl)-10-(1H-indol-3-ylmethyl)-16-(2-naphthalenylmethyl)-6,9,12,15,18,21,24,27-octaoxo-, (4R,10S,13S,16R,19S,22S,25S,28R)-
• AC-CYS-NLE-ARG-HIS-D-2-NAL-ARG-TRP-GLY-CYS-NH2 TRIFLUOROACETATE SALT
• HS024
• (4R,10S,13S,16R,19S,22S,25S,28R)-28-Acetamido-25-butyl-13,22-bis(3-carbamimidamidopropyl)-19-(1H-imidazol-4-ylmethyl)-10-(1H-indol-3-ylmethyl)-16-(2-naphthylmethyl)-6,9,12,15,18,21,24,27-octaoxo-1,2-dithia-5,8,11,14,17,20,23,26-octaazacyclononacosane-4-carboxamide
• AC-CYS-NLE-ARG-HIS-D-2-NAL-ARG-TRP-GLY-CYS-NH2