73734-07-3

• 常用中文名：4-(1H-苯并咪唑-2-基氨基)-1-哌啶羧酸乙酯
• 常用英文名：ethyl 4-(1H-benzimidazol-2-ylamino)piperidine-1-carboxylate
• CAS号：73734-07-3
• 分子式：C₁₅H₂₀N₄O₂
• 分子量：288.34500
• 发布时间：2018-11-24 11:19:18
• 更新时间：2025-09-25 20:40:18

名称

• 中文名: 4-(1H-苯并咪唑-2-基氨基)-1-哌啶羧酸乙酯
• 英文名: ethyl 4-(1H-benzimidazol-2-ylamino)piperidine-1-carboxylate
• 英文别名: EINECS 277-580-9; ethyl 4-(1H-benzo[d]imidazol-2-ylamino)piperidin-1-carboxylate; ethyl 4-[(3H-imidazo[4,5-b]pyridin-2-yl)amino]-1-piperdinecarboxylate; ethyl 4-(1H-benzimidazol-2-ylamino)-1-piperidine-carboxylate; 4-(1H-Benzimidazol-2-ylamino)-1-(ethoxycarbonyl)piperidine; (1H-benzimidazol-2-yl)-(1-ethoxycarbonyl-piperidin-4-yl)amine

物化性质

• 密度: 1.297g/cm3
• 沸点: 482.1ºC at 760 mmHg
• 分子式: C₁₅H₂₀N₄O₂
• 分子量: 288.34500
• 闪点: 245.4ºC
• 精确质量: 288.15900
• PSA: 73.48000
• LogP: 1.95550
• 折射率: 1.657

合成路线

73733-81-0 ~54% 73734-07-3

文献：Janssens; Torremans; Janssen; Stokbroekx; Luyckx Journal of Medicinal Chemistry, 1985 , vol. 28, # 12 p. 1925 - 1933

4857-06-1 58859-46-4 ~72% 73734-07-3

文献：Ishikawa, Minoru; Kubota, Dai; Yamamoto, Mikio; Kuroda, Chizuko; Iguchi, Maki; Koyanagi, Akihiro; Murakami, Shoichi; Ajito, Keiichi Bioorganic and Medicinal Chemistry, 2006 , vol. 14, # 7 p. 2109 - 2130

73733-81-0 74-88-4 ~28% 73734-07-3

文献：Janssen Pharmaceutica N.V. Patent: US4219559 A1, 1980 ;

58859-46-4 ~% 73734-07-3

文献：Janssens; Torremans; Janssen; Stokbroekx; Luyckx Journal of Medicinal Chemistry, 1985 , vol. 28, # 12 p. 1925 - 1933

73733-70-7 ~% 73734-07-3

文献：Janssens; Torremans; Janssen; Stokbroekx; Luyckx Journal of Medicinal Chemistry, 1985 , vol. 28, # 12 p. 1925 - 1933

4857-06-1 58859-46-4 497-19-8 ~% 73734-07-3

文献：Meiji Seika Kaisha, Ltd. Patent: US6420558 B1, 2002 ;

58859-46-4 208398-29-2 ~% 73734-07-3

文献：Hong, Yaping; Senanayake, Chris H.; Xiang, Tingjian; Vandenbossche, Charles P.; Tanoury, Gerald J.; Bakale, Roger P.; Wald, Stephen A. Tetrahedron Letters, 1998 , vol. 39, # 20 p. 3121 - 3124

4857-06-1 ~% 73734-07-3

文献：Hong, Yaping; Senanayake, Chris H.; Xiang, Tingjian; Vandenbossche, Charles P.; Tanoury, Gerald J.; Bakale, Roger P.; Wald, Stephen A. Tetrahedron Letters, 1998 , vol. 39, # 20 p. 3121 - 3124

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