1251765-07-7

• 常用中文名：替格瑞洛杂质 03
• 常用英文名：AR-C133913XX
• CAS号：1251765-07-7
• 分子式：C₁₄H₂₂N₆O₄S
• 分子量：370.427
• 发布时间：2018-06-22 21:07:38
• 更新时间：2025-08-25 11:20:02
• Ticagrelor metabolite M5, also known as AR-C133913XX, is a metabolite of Ticagrelor which is the first reversible oral P2Y12 receptor antagonist. Ticagrelor provides faster and more consistent ADP-receptor inhibition than Clopidogrel. Ticagrelor is used in the treatment of acute coronary syndromes (ACS).

名称

• 中文名: 替格瑞洛杂质 03
• 英文名: (1S,2S,3R,5S)-3-[7-Amino-5-(propylsulfanyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)-1,2-cyclopentanediol
• 英文别名: (1S,2S,3R,5S)-3-[7-Amino-5-(propylsulfanyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)-1,2-cyclopentanediol; 1,2-Cyclopentanediol, 3-[7-amino-5-(propylthio)-3H-1,2,3-triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)-, (1S,2S,3R,5S)-

物化性质

• 密度: 1.8±0.1 g/cm3
• 沸点: 711.4±70.0 °C at 760 mmHg
• 分子式: C₁₄H₂₂N₆O₄S
• 分子量: 370.427
• 闪点: 384.1±35.7 °C
• 精确质量: 370.142334
• LogP: -0.73
• 蒸汽压: 0.0±2.4 mmHg at 25°C
• 折射率: 1.787