常用名 | MS934 | CAS号 | 2756323-15-4 |
---|---|---|---|
价格 | ¥需询单/2mg ¥需询单/5mg ¥需询单/10mg | 纯度 | 98.0% |
备货期 | 10天 | 库存 | 现货 |
产品详情(用途,包装等)
用途: MS934 (MS-934) is a VHL-recruiting MEK1/2 degrader (PROTAC) with HT29 DC50 of 18/9 nM for MEK1/2 degradation, respectively.MS934 displays antiproliferation potency against HT29 cell with GI50 of 23 nM, degrades MEK1 and MEK2 and inhibits pMEK and pERK in a concentration-dependent manner in HT-29 and SK-MEL-28 cells. 物理化学性质: CAS号:2756323-15-4 常用中文名:MS934 常用英文名:MS934 分子式:C52H69F3In7O6S 分子量:1104.127 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |