| 常用名 | 5-([1,1'-联苯]-4-甲基)-N,N-二甲基-1H-四氮唑-1-甲酰胺 | CAS号 | 874902-19-9 |
|---|---|---|---|
| 价格 | 纯度 | 99.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: LY2183240 is a novel and highly potent blocker of anandamide uptake (IC50 = 270 pM). LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). IC50: 270 pM (anandamide uptake); 12.4 nM (FAAH)Target: FAAH; Anandamide uptakeFollowing i.p. administration in rats, LY2183240 increases brain anandamide concentration and exerts antinociceptive effects in formalin model of pain. 物理化学性质: CAS号:874902-19-9 常用中文名:5-([1,1'-联苯]-4-甲基)-N,N-二甲基-1H-四氮唑-1-甲酰胺 常用英文名:LY2183240 分子式:C17H17N5O 分子量:307.350 密度:1.2±0.1 g/cm3 沸点:506.1±53.0 °C at 760 mmHg 熔点:87-88ºC 闪点:259.9±30.9 °C 储存条件:2-8℃ |