| 常用名 | JNJ 10191584 马来酸盐 | CAS号 | 869497-75-6 |
|---|---|---|---|
| 价格 | 纯度 | 99.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: JNJ10191584 (VUF6002) maleate (compound 40) is an orally active and selective histamine H4 receptor antagonist with a Ki value of 26 nM. JNJ10191584 maleate shows 540-fold selectivity to H4 receptor over the H3 receptor with a Ki value of 14.1 μM. JNJ10191584 maleate inhibits chemotaxis of eosinophils and mast cells with IC50 values of 530 nM and 138 nM, respectively[1][2]. 物理化学性质: CAS号:869497-75-6 常用中文名:JNJ 10191584 马来酸盐 常用英文名:VUF6002 分子式:C17H19ClN4O5 分子量:394.81000 密度:N/A 沸点:461ºC at 760 mmHg 熔点:N/A 闪点:232.6ºC 储存条件:室温, 干燥 |