9,13B-二氢-1H-二苯并[c,f]咪唑并[1,5-a]氮杂卓-3-胺
更新时间：2025-09-06 17:36:51
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| 常用名 | 依匹斯汀 | CAS号 | 80012-43-7 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情（用途，包装等）
用途： Epinastine(WAL801) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Target: Histamine ReceptorEpinastine shows a high affinity to H1-receptors in receptor binding studies in the guinea pig ileum. Epinastine inhibits histamine-induced reactions in the skin or the lung of rats, dogs and guinea pigs [1]. Epinastine is able to displace specific [3H]NC-5Z binding at low concentrations in the locust nervous tissue. Epinastine binds to the honey bees neuronal octopamine receptor with Ki of 1.1 nM. Epinastine antagonises octopamine-induced cAMP formation in the insect brain [2]. Epinastine causes an inhibition of histamine release from rat peritoneal mast cells induced by both antigen-antibody reaction and compound 48/80. Epinastine is similarly effective in inhibiting compound 48/80-induced histamine release not only from isolated rat peritoneal mast cells but also from rat mesenterial pieces. Epinastine is effective in inhibiting not only Ca2+ uptake into lung mast cells in actively sensitized guinea pigs but also Ca2+ release from the intracellular Ca store of rat peritoneal mast cells exposed to both compound 48/80 and substance P [3]. Epinastine shows a dose- and time-dependent suppressive effect on IL-8, one of the chemokines for eosinophils, released from eosinophils isolated from atopic diseases [4]. 物理化学性质： CAS号：80012-43-7 常用中文名：依匹斯汀 常用英文名：Epinastine 分子式：C16H15N3 分子量：249.31000 密度：1.32 g/cm3 沸点：428ºC at 760 mmHg 熔点：270ºC 闪点：212.7ºC 储存条件：2-8℃ |
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- 产品名：9,13B-二氢-1H-二苯并[c,f]咪唑并[1,5-a]氮杂卓-3-胺
- 价格： ￥需询单/100mg ￥需询单/1g ￥需询单/250mg ￥需询单/50mg
- 纯度：98.0%
- 备货期：需询单
- 联系人：王汐瑶
- 上海化源世纪贸易有限公司
- 上海市 上海市 普陀区
- 产品名：9,13B-二氢-1H-二苯并[c,f]咪唑并[1,5-a]氮杂卓-3-胺
- 价格：
- 纯度：98.0%
- 备货期：10天
- 联系人：徐经理
- 广东翁江化学试剂有限公司
- 广东省 韶关市 翁源县
- 产品名：依匹斯汀
- 价格： ￥6400.0/500g
- 纯度：98.0%
- 备货期：需询单
- 联系人：朱丽丹
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参考价格：$106/10mM*1mLinDMSO