| 常用名 | UCSF924 | CAS号 | 1434515-70-4 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: UCSF924 is a potent and specific dopamine D4 receptor (DRD4) partial agonist with a EC50 of 4.2 nM. UCSF924 has a high-affinity with a Ki value of 3 nM for DRD4 and shows no measurable affinity for D2, D3 or the F261V/L328F D4 mutant. UCSF924 is a 7.4-fold bias toward arrestin over Gαi/o signaling, referenced to quinpirole[1]. 物理化学性质: CAS号:1434515-70-4 常用中文名:UCSF924 常用英文名:UCSF924 分子式:C20H22N2O2 分子量:322.40 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |