常用名 | GSK-199 hydrochloride | CAS号 | 1549811-53-1 |
---|---|---|---|
价格 | ¥需询单/1g ¥需询单/5g | 纯度 | 98.0% |
备货期 | 需询单 | 库存 | 现货 |
产品详情(用途,包装等)
用途: GSK-199 hydrochloride is a potent, highly selective and reversible protein arginine deiminase PAD4 inhibitor with IC50 of 250 nM in FP binding assay (0.2 mM Ca), 200 nM in PAD4 NH3 release inhibition assay; shows high specificity for PAD4 over PAD1/2/3/6; affects cellular citrullination and mimic the deficiency in NET production in mice; significantly decreases in complement C3 deposition in both synovium and cartilage in mice. 物理化学性质: CAS号:1549811-53-1 常用中文名:GSK-199 hydrochloride 常用英文名:GSK-199 hydrochloride 分子式:C24H29ClN6O2 分子量:468.979 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:-20°C,密闭,干燥 |