| 常用名 | MRK-016 | CAS号 | 342652-67-9 |
|---|---|---|---|
| 价格 | ¥9600.0/50mg ¥需询单/1g ¥需询单/1g ¥需询单/1g | 纯度 | 98.0% |
| 备货期 | 1天 | 库存 | 现货 |
| 产品网页 | http://www.aladdin-e.com/zh_cn/M286670.html | ||
| 产品详情(用途,包装等)
用途: MRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77 and 1.4 nM for human GABAA α1β3γ2, GABAA α2β3γ2, GABAA α3β3γ2, and GABAA α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 物理化学性质: CAS号:342652-67-9 常用中文名:MRK-016 常用英文名:MRK 016 分子式:C17H20N8O2 分子量:368.39 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:2-8℃ |