| 常用名 | 4,6-二(苯甲酰氨基)-1,3-苯二羧酸 | CAS号 | 70553-45-6 |
|---|---|---|---|
| 价格 | $需询单/100mg $需询单/250mg $需询单/500mg | 纯度 | 98.0% |
| 备货期 | 3天 | 库存 | 3 |
| 产品网页 | https://www.dcchemicals.com/product_show-NS3763.html | ||
| 产品详情(用途,包装等)
NS3763 is a noncompetitive antagonist of GLUK5 receptor. NS3763 displays selectivity for inhibition of domoate-induced increase in intracellular calcium mediated through the GLU(K5) subtype (IC(50) = 1.6 microM) of kainate receptors compared with the GLU(K6) subtype (IC(50) > 30 microM). NS3763 inhibits the GLU(K5)-mediated response in a noncompetitive manner. NS3763 selectively inhibits l-glutamate- and domoate-evoked currents through GLU(K5) receptors in HEK293 cells. |