Journal of Organic Chemistry 2008-08-15

Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid.

Sébastien Bénard, Luc Neuville, Jieping Zhu

文献索引：J. Org. Chem. 73 , 6441, (2008)

摘要

Reaction of azoles, amides, and sulfonamides in dichloroethane with readily available cyclopropylboronic acid in the presence of copper acetate and sodium carbonate afforded the N-cyclopropyl derivatives in good to excellent yields.

结构式	名称/CAS号	分子式	全部文献
	环丙基硼酸 CAS:411235-57-9	C₃H₇BO₂

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Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid.

摘要

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