… -activity relationships of 1, 4-dihydro-(1H, 4H)-quinoxaline-2, 3-diones as N-methyl-D-aspartate (glycine site) receptor antagonists. 1. Heterocyclic substituted 5-alkyl …

MJ Fray, DJ Bull, CL Carr, ECL Gautier…

文献索引：Abenhaim, David; Diez-Barra, Enrique; Hoz, Antonio de la; Loupy, Andre; Sanchez-Migallon, Ana Heterocycles, 1994 , vol. 38, # 4 p. 793 - 802

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被引用次数: 57

摘要

... Binding affinity increased significantly if the heterocyclic group, eg 1,2,3-triazol-1-yl ... compounds (1−17) (Chart 2) in which the hydrogen bond acceptor is an aromatic heterocycle. ... were most conveniently prepared by reaction of the benzylic bromide 35 with heterocycles such as ...

~70%

~0%

详细

Synthesis and structure–activity relationship of 1-and 2-sub...

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An investigation into the alkylation of 1, 2, 4-triazole

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Synthesis of 1-alkyl-1, 2, 4-triazoles: a new one-pot regios...

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Etude dans la serie des organosilylazoles: I. Action des hal...

[Gasparini, J. P.; Gassend, R.; Maire, J. C.; Elguero, J. Journal of Organometallic Chemistry, 1980 , vol. 188, # 2 p. 141 - 150]

N-Alkylation of amines with alcohols over nanosized zeolite ...

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