2', 6'-Dimethylphenoxyacetyl: A New Achiral High Affinity P3-P2 Ligand for Peptidomimetic-Based HIV Protease Inhibitors

…, C Grand-Maître, D Lamarre, F Liard…

文献索引：Moreau,C.; Rouessac,F. Bulletin de la Societe Chimique de France, 1973 , p. 3427 - 3432

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被引用次数: 35

摘要

... One notable exception is the 3-hydroxy-2-methylbenzoyl moiety (7) found in inhibitors such as Viracept (nelfinavir, AG 1343) 10a,b and the closely related LY316340, 10c and some C 2 symmetric inhibitors. 10d A common feature of P 3 -P 2 ligands introduced to date is the ...