Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores

R Betageri, T Gilmore, D Kuzmich, TM Kirrane…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 22 p. 6842 - 6851

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被引用次数: 8

摘要

... Bioorganic & Medicinal Chemistry Letters. ... a Department of Medicinal Chemistry, Boehringer Ingelheim ... The glucocorticoid receptor (GR), a member of the nuclear receptor family, is an attractive drug discovery target, and chemical entities that function as GR agonists and ...