NGB 2904 and NGB 2849: two highly selective dopamine D 3 receptor antagonists

J Yuan, X Chen, R Brodbeck, R Primus, J Braun…

文献索引：Yuan, Jun; Chen, Xi; Brodbeck, Robbin; Primus, Renee; Braun, Julia; Wasley, Jan W. F.; Thurkauf, Andrew Bioorganic and Medicinal Chemistry Letters, 1998 , vol. 8, # 19 p. 2715 - 2718

全文：HTML全文

被引用次数: 87

摘要

N-(4-[4-{2, 3-dichlorophenyl}-1-piperazinyl] butyl)-3-fluorenylcarboxamide and N-(4-[4-{2, 3- dichlorophenyl}-1-piperazinyl] butyl)-2-biphenylenylcarboxamide were prepared in several steps from 2, 3-dichloroaniline. These compounds were identified as highly selective dopamine D3 receptor antagonists.