Tetrahedron Letters

Synthesis of amide libraries with immobilized HOBt

S Vokkaliga, J Jeong, WR LaCourse, A Kalivretenos

文献索引：Vokkaliga, Smitha; Jeong, Jeannie; Lacourse, William R.; Kalivretenos, Aristotle Tetrahedron Letters, 2011 , vol. 52, # 21 p. 2722 - 2724

全文：HTML全文

被引用次数: 8

摘要

Abstract Highly reactive N-acylating solid-phase reagents based on macroporous polystyrene-bound 1-hydroxybenzotriazole (P-HOBt) and silica-bound 1- hydroxybenzotriazole (Si-HOBt) were prepared and compared for reactivity by synthesis of small combinatorial libraries of acetamides and benzamides.