Archiv der Pharmazie

A Simple Procedure for Synthesis of Roxindole, a Dopamine D2??Receptor Agonist

F Csende

文献索引：Csende, Ferenc Archiv der Pharmazie (Weinheim, Germany), 2001 , vol. 334, # 7 p. 253 - 254

全文：HTML全文

被引用次数: 1

摘要

Abstract A modified convenient and high yielding synthetic route for the preparation of the dopamine agonist roxindole 1 is described. The key step in our method is the phase-transfer catalyzed reaction of γ-butyrolactone with 5-methoxyindole which results in the indolyl-