Organic letters

Selective deprotection of methanesulfonamides to amines

H Naito, T Hata, H Urabe

文献索引：Naito, Hiroyuki; Hata, Takeshi; Urabe, Hirokazu Organic Letters, 2010 , vol. 12, # 6 p. 1228 - 1230

全文：HTML全文

被引用次数: 11

摘要

Sulfonamides are a stable derivative of amines, and they are frequently used as versatile intermediates and for the protection of amines in organic synthesis. However, their stability is not without its drawbacks, because once their deprotection giving back to the parent amines is desired, available methods are limited and often require harsh conditions.(1) To circumvent this problem, new sulfonamides carrying an extra functional group that facilitates the release of the amine portion have ...