Tetrahedron

Iodine-induced regioselective direct alkylation of azoles via in situ formed alkyliodide

W Chen, R Yan, D Tang, S Guo, X Meng, B Chen

文献索引：Chen, Wenlin; Yan, Rulong; Tang, Dong; Guo, Shuaibo; Meng, Xu; Chen, Baohua Tetrahedron, 2012 , vol. 68, # 38 p. 7956 - 7959

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被引用次数: 5

摘要

We have developed an efficient, metal-free, convenient and relatively cheap method for iodine-induced direct alkylation of azoles via in situ formed alkyliodide. A series of heterocyclic derivatives are readily prepared under mild conditions in moderate to good yields and high regioselectivity.