Synthesis of N-protected erythro-phenylalanylepoxides

…, G Raidaru, K Linask, J Järv, M Zetterström…

文献索引：Heinsoo; Raidaru; Linask; Jarv; Zetterstrom; Langel Tetrahedron Asymmetry, 1995 , vol. 6, # 9 p. 2245 - 2247

被引用次数: 23

摘要

N-et-Protected amino epoxides of general formula (6) are potential building blocks for synthesis of hydroxyethylene dipeptide isomers 1.2.3. These amino acid derivatives contain two stereogenic centers, which have been found to be important for their biological activity, but complicate chemical synthesis of these compounds. Stereoselective synthesis of erythro-isomers of several Cbz-N-et-protected ot - amino epoxides has been described recently 4. Supplementary to ...

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