Simple, efficient catalyst system for the palladium-catalyzed amination of aryl chlorides, bromides, and triflates

JP Wolfe, H Tomori, JP Sadighi, J Yin…

文献索引：Grigg, Ronald; Mitchell, Thomas R.B.; Tongpenyai, Ngampong Synthesis, 1981 , # 6 p. 442 - 444

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被引用次数: 790

摘要

... 1 and 2 (Figure 1). 2e However, the preparation of these phosphines required a multistep synthesis. ... 4-chlorotoluene gave higher yields than were obtained with 3 or 4 (entry 6); use of ... diaryl products were typically ∼10−20/1 for reactions of primary amines with p-substituted aryl ...