CsF–Celite catalyzed facile N-alkylation of 2 (3H)-benzoxazolones and antimicrobial properties of 2-substituted benzoxazole and 3-substituted-2 (3H)-benzoxazolone …

…, RV Rao, JS Yadav, USN Murty, KP Kumar

文献索引：Murty; Ram, Kesur R.; Rao, Rayudu Venkateswara; Yadav; Kumar, K. Pranay Medicinal Chemistry Research, 2011 , vol. 20, # 5 p. 626 - 636

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被引用次数: 9

摘要

Abstract The synthesis and antimicrobial activity studies of a new series of cyclic amine containing benzoxazoles and benzoxazolone-2 (3 H)-ones derivatives were described. The alkylation of benzoxazolone was carried out using cesium fluoride–Celite. The newly synthesized compounds with the influence of the induction of the cyclic amine moiety in the benzoxazole scaffold have been evaluated with respect to the antibacterial and antifungal ...