Tetrahedron: Asymmetry

Enantioselective benzoylation of racemic amines using chiral benzimidazolide as a benzoylating agent

AV Karnik, SS Kamath

文献索引：Karnik, Anil V.; Kamath, Suchitra S. Tetrahedron Asymmetry, 2008 , vol. 19, # 1 p. 45 - 48

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被引用次数: 38

摘要

Enantioselective acylation/kinetic resolution of racemic amines has been achieved by using a chiral benzimidazolide, namely,(S)-1-benzoyl-2-(α-acetoxyethyl) benzimidazole 2. This nonenzymatic acylating reagent requires mild reaction conditions and proceeds with good ...