[(3-Chlorophenyl) piperazinylpropyl] pyridazinones and analogues as potent antinociceptive agents

MP Giovannoni, C Vergelli, C Ghelardini…

文献索引：Journal of Medicinal Chemistry, , vol. 46, # 6 p. 1055 - 1059

被引用次数: 83

摘要

... Journal of Medicinal Chemistry. ... Chemistry. The synthetic pathway affording the final 5−8 is depicted in Scheme 1. With the exception of 3c and 4c, the isoxazoles 3 and the isoxazolo[3,4-d]pyridazinones 4 were previously described. ...

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Base??and Copper??Catalysed Condensation of Primary Activate...

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