Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists

S Sasmal, G Balaji, HRK Reddy…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 22, # 9 p. 3157 - 3162

被引用次数: 33

摘要

... Bioorganic & Medicinal Chemistry Letters. ... As will become apparent we lost in affinity for the MCH1 receptor by this scaffold switch which called for additional SAR explorations of the eastern side chain that are described in this Letter leading up to a molecule with good efficacy ...

3612-20-2

N-苄基-4-哌啶酮

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