Tetrahedron letters

Amino protection using triazones

S Knapp, JJ Hale, M Bastos, FS Gibson

文献索引：Knapp, Spencer; Hale, Jeffrey J.; Bastos, Margarita; Gibson, Frank S. Tetrahedron Letters, 1990 , vol. 31, # 15 p. 2109 - 2112

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被引用次数: 43

摘要

Abstract Primary amines protected by incorporation into a “triazone” derivative (3) are stable to various reduction, oxidation, organometallic, and basic hydrolysis conditions, and may be regenerated by treatment with aqueous ammonium chloride at 70. An application to polyamine synthesis is described.