Enantiomerically Pure Cyclopropylamines from Cyclopropylboronic Esters

J Pietruszka, G Solduga

文献索引：Pietruszka, Joerg; Solduga, Gemma European Journal of Organic Chemistry, 2009 , # 34 p. 5998 - 6008

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被引用次数: 0

摘要

Abstract Cyclopropylamines are versatile intermediates and products both in organic synthesis in general and for active substances in particular. Although the synthesis of the corresponding enantiomerically pure cyclopropylboronic esters had been established previously, the C–B to C–N transformation was elusive. A detailed study directed towards the synthesis of several enantiomerically pure cyclopropylamines is disclosed; ...