Tetrahedron Letters

A mild Boc deprotection and the importance of a free carboxylate

A Thaqi, A McCluskey, JL Scott

文献索引：Thaqi, Ali; McCluskey, Adam; Scott, Janet L. Tetrahedron Letters, 2008 , vol. 49, # 49 p. 6962 - 6964

被引用次数: 23

摘要

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... We report a facile and rapid removal of Boc protecting groups using microwave heating in H 2 O, with deprotection only requiring a free carboxylic acid group in the starting material. Unlike previous approaches, no additional reagents are required. ... Boc-deprotection of substances ...

~99%

~98%

4353-32-6

N'-对甲苯磺酰基-L-精氨酸

~97%

~60%

~0%

~99%

~99%

~99%

~92%

~29%

~98%

~99%

~94%

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