SUVN-502
Names
[ CAS No. ]:
701205-60-9
[ Name ]:
SUVN-502
Biological Activity
[Description]:
Masupirdine free base (SUVN-502 free base) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine free base (SUVN-502 free base) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease[1].
[Related Catalog]:
[Target]
Ki: 2.04 nM (human 5-HT6 receptor)[1]
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C21H24BrN3O3S
[ Molecular Weight ]:
478.40