SUVN-502 mesylate
Names
[ CAS No. ]:
1791396-46-7
[ Name ]:
SUVN-502 mesylate
Biological Activity
[Description]:
Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease[1].
[Related Catalog]:
[Target]
5-HT6 Receptor:2.04 nM (Ki)
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C23H32BrN3O9S3
[ Molecular Weight ]:
670.61