ENMD 547

Names

[ Name ]:
ENMD 547

[Synonym ]:
enmd 547

Biological Activity

[Description]:

ENMD-1068 hydrobromide is a potent PAR2 antagonist. ENMD-1068 hydrobromide attenuates joint inflammation in a dose-dependent manner. ENMD-1068 hydrobromide can be used in research of joint inflammation[1].

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Protease-Activated Receptor (PAR)

Research Areas >> Inflammation/Immunology

[References]

[1]. Kelso EB, et, al. Therapeutic promise of proteinase-activated receptor-2 antagonism in joint inflammation. J Pharmacol Exp Ther. 2006 Mar;316(3):1017-24.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₅H₃₀BrN₃O₂

[ Molecular Weight ]:
364.32

[ Exact Mass ]:
363.15200

[ PSA ]:
66.64000

[ LogP ]:
2.75660

Related Compounds

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