644961-61-5

644961-61-5 structure

Name: ENMD 547
Chemical Name: 6-amino-1-[4-(3-methylbutanoyl)piperazin-1-yl]hexan-1-one,hydrobromide
CAS Number: 644961-61-5
Molecular Formula: C₁₅H₃₀BrN₃O₂
Molecular Weight: 364.32
Catalog: Signaling Pathways GPCR/G Protein Protease-Activated Receptor (PAR)
Create Date: 2017-01-28 20:38:32
Modify Date: 2025-10-19 18:10:49
ENMD-1068 hydrobromide is a potent PAR2 antagonist. ENMD-1068 hydrobromide attenuates joint inflammation in a dose-dependent manner. ENMD-1068 hydrobromide can be used in research of joint inflammation[1].

Name	6-amino-1-[4-(3-methylbutanoyl)piperazin-1-yl]hexan-1-one,hydrobromide
Synonyms	enmd 547

Description	ENMD-1068 hydrobromide is a potent PAR2 antagonist. ENMD-1068 hydrobromide attenuates joint inflammation in a dose-dependent manner. ENMD-1068 hydrobromide can be used in research of joint inflammation[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Protease-Activated Receptor (PAR) Research Areas >> Inflammation/Immunology
References	[1]. Kelso EB, et, al. Therapeutic promise of proteinase-activated receptor-2 antagonism in joint inflammation. J Pharmacol Exp Ther. 2006 Mar;316(3):1017-24.