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EGFR-IN-25

Names

[ CAS No. ]:
2749562-63-6

[ Name ]:
EGFR-IN-25

Biological Activity

[Description]:

EGFR-IN-25 is a potent EGFR inhibitor with IC50s of 9 nM and 60 nM for BaF3 cells (EGFR DEL19/T790M/C797S) and A431 cells (WT), respectively[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> JAK/STAT Signaling >> EGFR
Signaling Pathways >> Protein Tyrosine Kinase/RTK >> EGFR

[References]

[1]. New pyrazine compound. WO2021244505A1.

Chemical & Physical Properties

[ Molecular Formula ]:
C34H43N9O2

[ Molecular Weight ]:
609.76


Related Compounds