Difelikefalin HCl

Names

[ Name ]:
Difelikefalin HCl

Biological Activity

[Description]:

Difelikefalin is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin is selective for KOR over the μ-opioid receptor.

Chemical & Physical Properties

[ Molecular Formula ]:
C₃₆H₅₆Cl₃N₇O₆

[ Molecular Weight ]:
789.237

Related Compounds

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.