AZ-8838

Names

[ Name ]:
AZ-8838

Biological Activity

[Description]:

AZ-8838 (AZ8838) is a potent, and selective PAR2 antagonist with Kd of 125 nM; shows excellent selectivity over PAR1 and PAR4 (>50 uM).

[References]

References 1. Cheng RKY, et al. Nature. 2017 May 4;545(7652):112-115. View Related Products by Target Protease-activated Receptor (PAR)

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₃H₁₅FN₂O

[ Molecular Weight ]:
234.274

Related Compounds

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.