Dual DRAK1 and DRAK2 inhibitor 1

Names

[ Name ]:
Dual DRAK1 and DRAK2 inhibitor 1

Biological Activity

[Description]:

Dual DRAK1 and DRAK2 inhibitor 1 is a potent, dual DRAK2/1 inhibitor Kd value of 9/5 nM, respectively;Dual DRAK1 and DRAK2 inhibitor 1 also is a functional inhibitor of DRAK2/1 enzymatic activity with IC50 of 0.86 and 2.25 uM.Dual DRAK1 and DRAK2 inhibitor 1 is a chemical tool compound to study DRAK1 and DRAK2 biology.

[References]

1. Ling-Jie Gao, et al. J Med Chem. 2014 Sep 25;57(18):7624-43.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₂H₂₄N₂O₃S

[ Molecular Weight ]:
396.505

Related Compounds

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