Name | Dual DRAK1 and DRAK2 inhibitor 1 |
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Description | Dual DRAK1 and DRAK2 inhibitor 1 is a potent, dual DRAK2/1 inhibitor Kd value of 9/5 nM, respectively;Dual DRAK1 and DRAK2 inhibitor 1 also is a functional inhibitor of DRAK2/1 enzymatic activity with IC50 of 0.86 and 2.25 uM.Dual DRAK1 and DRAK2 inhibitor 1 is a chemical tool compound to study DRAK1 and DRAK2 biology. |
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References | 1. Ling-Jie Gao, et al. J Med Chem. 2014 Sep 25;57(18):7624-43. |
Molecular Formula | C22H24N2O3S |
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Molecular Weight | 396.505 |